MERCK SHARP & DOHME B.V.

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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology Matters Rank in Class
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 97158
 
 
 
C07D HETEROCYCLIC COMPOUNDS 7292
 
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 1085
 
 
 
C07K PEPTIDES 10126
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 940
 
 
 
C07J STEROIDS811
 
 
 
A61F FILTERS IMPLANTABLE INTO BLOOD VESSELS; PROSTHESES; DEVICES PROVIDING PATENCY TO, OR PREVENTING COLLAPSING OF, TUBULAR STRUCTURES OF THE BODY, E.G. STENTS; ORTHOPAEDIC, NURSING OR CONTRACEPTIVE DEVICES; FOMENTATION; TREATMENT OR PROTECTION OF EYES OR EARS; BANDAGES, DRESSINGS OR ABSORBENT PADS; FIRST-AID KITS 7133
 
 
 
A61M DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY 5149
 
 
 
C12N MICRO-ORGANISMS OR ENZYMES; COMPOSITIONS THEREOF 5162
 
 
 
C12P FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE 594

Top Patents (by citation)

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Recent Publications

Publication # Title Filing Date Pub Date Intl Class
2017/0202,209 APPARATUS AND METHOD FOR PRESERVING MUCOSAFeb 25, 16Jul 20, 17[A01N, C08B, B01F, A61L, A22B]

Recent Patents

Patent # Title Filing Date Issue Date Intl Class
9884043 RORgammaT inhibitorsMar 20, 17Feb 06, 18[A61K, C07D]
9834605 Antibodies to human programmed death receptor PD-1Dec 19, 14Dec 05, 17[G01N, C07K]
9820973 Pharmaceutical formulation comprising losartan potassium and chlorthalidoneNov 24, 14Nov 21, 17[A61K]
9790226 4-imidazopyridazin-1-yl-benzamides and 4-imidazotriazin-1-yl-benzamides as BtK inhibitorsFeb 09, 16Oct 17, 17[A61K, C07D]
9757552 Applicator for inserting an implantJan 20, 06Sep 12, 17[A61M]
9758524 4-imidazopyridazin-1-yl-benzamides as Btk inhibitorsFeb 09, 16Sep 12, 17[A61K, C07D]
9718828 BTK InhibitorsAug 30, 16Aug 01, 17[A61K, C07D, A61P]
9603838 RORgammaT inhibitorsJun 26, 15Mar 28, 17[A61K, C07D]
9540361 N-substituted azetidine derivativesDec 16, 11Jan 10, 17[C07D]
9464108 Combined synthesis route for desogestrel and etonogestrelMar 13, 13Oct 11, 16[C07J]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2016/0159,800 MK2 INHIBITORSAbandonedJul 09, 15Jun 09, 16[C07D]
2014/0296,833 INTRAUTERINE SYSTEM FOR USE IN MEDICAL TREATMENTAbandonedNov 06, 13Oct 02, 14[A61M]
2014/0221,333 BTK INHIBITORSAbandonedJul 19, 12Aug 07, 14[A61K, C07D]
2014/0155,406 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDES AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDES BTK INHIBITORSAbandonedJul 11, 12Jun 05, 14[A61K, C07D]
2014/0056,962 DRUG DELIVERY SYSTEMAbandonedOct 31, 13Feb 27, 14[A61K]
8575152 Non-steroidal compounds useful as glucocorticoid receptor modulatorsExpiredAug 25, 06Nov 05, 13[A61K, C07D, A61P]
2013/0272,956 (11beta, 17alpha)-11-(4-(2-11C-ACETYL)PHENYL)-17,23-EPOXY-19,24-DINORCHOLA-4,9,20-TRIEN-3-ONEAbandonedJun 17, 11Oct 17, 13[A61K, C07J]
2013/0150,337 SUBSTITUTED 16,17-ANNELLATED STEROID COMPOUNDS FOR USE IN WOMENS HEALTHAbandonedFeb 05, 13Jun 13, 13[C07J]
2013/0131,029 ANTISOLVENT SOLIDIFICATION PROCESSAbandonedJan 09, 13May 23, 13[A61K, B01D, C07J, C01D]
2013/0106,013 METHOD FOR DOSING A FLUID FORMULATION CONTAINING A MEDICINAL SUBSTANCEAbandonedJul 05, 11May 02, 13[A61J]
2013/0014,763 INTRAUTERINE DEPOSITAbandonedSep 18, 12Jan 17, 13[A61F, B29C]
2012/0302,552 S-MIRTAZAPINE FOR THE TREATMENT OF HOT FLUSHAbandonedAug 09, 12Nov 29, 12[A61K, A61P]
8299091 Aminoisoquinoline thrombin inhibitor with improved bioavailabilityExpiredAug 06, 07Oct 30, 12[A61K, C07D]
2012/0258,957 HETEROCYCLIC DERIVATIVESAbandonedNov 22, 10Oct 11, 12[A61K, C07D, A61P]
2012/0231,497 SELECTIVE ENZYMATIC HYDROLYSIS OF C-TERMINAL TERT-BUTYL ESTERS OF PEPTIDESAbandonedMay 17, 12Sep 13, 12[C12P, C07K]
8211927 5-phenyl-isoxazole-3-carboxamide derivatives as TRPV1 modulatorsExpiredJul 31, 08Jul 03, 12[A61K, C07D]
2012/0095,002 ISOXAZOLE-5-CARBOXAMIDE DERIVATIVESAbandonedFeb 02, 10Apr 19, 12[A61K, C07D, A61P]
8143246 1-(4-(pyridin-2-yl)benzyl)imidazolidine-2,4-dione derivativesExpiredFeb 15, 10Mar 27, 12[A61K, C07D]
2012/0071,481 ISOXAZOLE-5-CARBOXAMIDE DERIVATIVESAbandonedFeb 02, 10Mar 22, 12[A61K, C07D, A61P]
8133885 Non steroidal glucocorticoid receptor modulatorsExpiredFeb 14, 06Mar 13, 12[A61K, C07D, A61P]

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